Hubei Honest Biochemical Co., Ltd.

Product Name: Tianeptine sodium salt

Synonyms: TIANEPTINE SODIUM;TIANEPTINE SODIUM SALT;7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide Sodium Salt;S-1574;Stablon;7-[(3-chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepine-11-yl)amino]heptanoic acid s,s dioxide sodium salt;[7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepine 5,5-dioxide)-11-ylamino]heptanoic acid]sodium salt;3-Chloro-6,11-dihydro-6-methyl-11-[6-(sodiooxycarbonyl)hexylamino]dibenzo[c,f][1,2]thiazepine 5,5-dioxide

CAS: 30123-17-2

MF: C21H24ClN2NaO4S

MW: 458.93

EINECS: 250-059-3

 

Sodium Tianeptin salt is a salt of Tianeptin. Tianeptin, a tricyclic compound, is a selective facilitator of 5-HT (serotonin;sc-201146) uptake in vitro and in vivo. Additionally, Tianeptin is reported to act as a selective inhibitor of dopamine uptake .Tianeptin does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptin was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptin in vitro .The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation.